Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM83506 ((5Z)-5-[[2-(3-isopropoxypropylamino)-4-keto-9-meth...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Burnham Center for Chemical Genomics Curated by PubChem BioAssay | Assay Description Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford Burnham Medical Research Institute (SBMRI, La Jolla, CA... | PubChem Bioassay (2012) BindingDB Entry DOI: 10.7270/Q2PC30Z9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401033 (US10005735, Compound 31) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264417 (CHEMBL4104719) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264415 (CHEMBL4096289) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <200 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401008 (US10005735, Compound 17) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <200 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264457 (CHEMBL4080490) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <200 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401006 (US10005735, Compound 15) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401020 (US10005735, Compound 19) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <200 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM400998 (US10005735, Compound 11) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264482 (CHEMBL4086748) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >300 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in beta5 inhibitor MG132 pretreated human HeLa cells expressing UbG76... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264420 (CHEMBL4100384) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM224012 (Capzimin | US10005735, Compound 12) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM224012 (Capzimin | US10005735, Compound 12) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 340 | n/a | n/a | n/a | n/a | 7.5 | 30 |
California Institute of Technology | Assay Description Fluorescence polarization assays were performed in low-volume 384-well solid black plates (Molecular Devices) in quadruplicate. The assays were perfo... | Nat Chem Biol 13: 486-493 (2017) Article DOI: 10.1038/nchembio.2326 BindingDB Entry DOI: 10.7270/Q24J0D0B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264419 (CHEMBL4073553) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 390 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401034 (US10005735, Compound 32) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264515 (CHEMBL4070821) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM400992 (US10005735, Compound 5) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM400996 (US10005735, Compound 9) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401029 (US10005735, Compound 27) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264471 (CHEMBL4093962) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264419 (CHEMBL4073553) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in beta5 inhibitor MG132 pretreated human HeLa cells expressing UbG76... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM88892 (MLS000401485 | N-(2-chlorophenyl)-2-[(2E)-2-[(2-mo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 658 | n/a | n/a | n/a | n/a | n/a | n/a |
Burnham Center for Chemical Genomics Curated by PubChem BioAssay | Assay Description Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford Burnham Medical Research Institute (SBMRI, La Jolla, CA... | PubChem Bioassay (2012) BindingDB Entry DOI: 10.7270/Q2PC30Z9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401030 (US10005735, Compound 28) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401009 (US10005735, Compound 18) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401026 (US10005735, Compound 24) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM39775 ((5E)-5-[(E)-3-[4-(dimethylamino)phenyl]prop-2-enyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 703 | n/a | n/a | n/a | n/a | n/a | n/a |
Burnham Center for Chemical Genomics Curated by PubChem BioAssay | Assay Description Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford Burnham Medical Research Institute (SBMRI, La Jolla, CA... | PubChem Bioassay (2012) BindingDB Entry DOI: 10.7270/Q2PC30Z9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM46229 (4-chloranyl-N-(3,4-dihydro-2H-thiochromen-4-yl)-3-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 763 | n/a | n/a | n/a | n/a | n/a | n/a |
Burnham Center for Chemical Genomics Curated by PubChem BioAssay | Assay Description Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford Burnham Medical Research Institute (SBMRI, La Jolla, CA... | PubChem Bioassay (2012) BindingDB Entry DOI: 10.7270/Q2PC30Z9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM4314 ((2E)-2-(2,3-dihydro-1H-indol-1-ylcarbonyl)-3-(3,4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 798 | n/a | n/a | n/a | n/a | n/a | n/a |
Burnham Center for Chemical Genomics Curated by PubChem BioAssay | Assay Description Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford Burnham Medical Research Institute (SBMRI, La Jolla, CA... | PubChem Bioassay (2012) BindingDB Entry DOI: 10.7270/Q2PC30Z9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM400995 (US10005735, Compound 8) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264483 (CHEMBL4105598) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264416 (CHEMBL4069023) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264453 (CHEMBL4088568) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401023 (US10005735, Compound 21) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401021 (US10005735, Compound 20) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264426 (CHEMBL4095913) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264526 (CHEMBL4093473) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264491 (CHEMBL4101230) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264455 (CHEMBL4060337) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM400994 (US10005735, Compound 7) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM88971 ((2E)-2-[(2Z)-2-(3-bromanyl-5-methoxy-4-oxidanylide...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 914 | n/a | n/a | n/a | n/a | n/a | n/a |
Burnham Center for Chemical Genomics Curated by PubChem BioAssay | Assay Description Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford Burnham Medical Research Institute (SBMRI, La Jolla, CA... | PubChem Bioassay (2012) BindingDB Entry DOI: 10.7270/Q2PC30Z9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401028 (US10005735, Compound 26) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264426 (CHEMBL4095913) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in beta5 inhibitor MG132 pretreated human HeLa cells expressing UbG76... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264422 (CHEMBL4091693) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in beta5 inhibitor MG132 pretreated human HeLa cells expressing UbG76... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264424 (CHEMBL4078891) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264518 (CHEMBL4087722) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM50264547 (CHEMBL4077883) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California San Diego Curated by ChEMBL | Assay Description Inhibition of 26S proteasome regulatory subunit RPN11 deubiquitinating activity in human erythrocytes using Ub4-pepOG protein substrate preincubated ... | J Med Chem 60: 1343-1361 (2017) Article DOI: 10.1021/acs.jmedchem.6b01379 BindingDB Entry DOI: 10.7270/Q22F7QX5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM400988 (US10005735, Compound 1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM88962 ((6R,7R)-7-[[(2E)-2-(2-amino-1,3-thiazol-4-yl)-2-(c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 1.04E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Burnham Center for Chemical Genomics Curated by PubChem BioAssay | Assay Description Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford Burnham Medical Research Institute (SBMRI, La Jolla, CA... | PubChem Bioassay (2012) BindingDB Entry DOI: 10.7270/Q2PC30Z9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401031 (US10005735, Compound 29) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
26S proteasome non-ATPase regulatory subunit 14 (Homo sapiens (Human)) | BDBM401007 (US10005735, Compound 16) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research | Assay Description In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i... | Bioorg Med Chem 17: 8086-92 (2009) BindingDB Entry DOI: 10.7270/Q22R3V09 | |||||||||||
More data for this Ligand-Target Pair |
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